BIT's 16th Annual Congress of International Drug Discovery Science and Technology-2018
Scientific Program
 
BIT's 16th Annual Congress of International Drug Discovery Science and Technology-2018
Theme: Rethinking the Next Big Things in Pharma Innovations
Time: August 16-19, 2018 
Place: Boston Marriott Cambridge, USA
 
Scientific Program
Stream 1 Stream 2 Stream 3 Stream 4 Stream 5

 

Stream 3: Industrial Art Gallery
-Arts in Billion Dollar Molecules and Next Generation Therapy

Substream 3-1: Improved Linear Drug Discovery on Selected Current Drug Targets
Substream 3-2: Novel Small Molecule Inhibitors and Agonists
Substream 3-3: Follow-on Drugs and Repositioning Drug Discovery
Substream 3-4: Novel Biotherapeutic Discovery
Substream 3-5: Smart DDS and Nanomedicine

Substream 3-6: Clinical Trial Gateway and Translational Convergence

Substream 3-7: Arts of Next Generation Therapy

 

 

Substream 3-2: Novel Small Molecule Agonists and Inhibitors
 

Session 3201: Novel Small Molecule Agonists and Inhibitors

Day 1: Afternoon, Thursday, August 16, 2018

Place: Concept Room, 2nd Floor

13:30-17:10

Chair: Dr. Wei-Sheng Huang, Senior Director, Theseus Pharmaceuticals, USA
Co-Chair: Dr. Alexei G. Basnakian, Professor, University of Arkansas for Medical Sciences, USA
Time FaceOn Speeches and Speakers
13:30-13:35 Chair's Introduction
13:35-13:55

Title: Tackling Mutation-based Resistance in Kinase Drug Discovery: Brigatinib and AP32788

Dr. Wei-Sheng Huang, Senior Director, Theseus Pharmaceuticals, USA
13:55-14:15

Title: The Role of F11R Antagonists in Neointimal Hyperplasia in Dialysis Vascular Accesses

Dr. Moro O. Salifu, Chair, Department of Medicine; Chief, Division of Nephrology, State University of New York Downstate Medical Center, USA

14:15-14:35

Title: Discovering Drug Leads by Practical NMR Strategies

Dr. Steven LaPlante, Professor, University of Quebec INRS-IAF; Founder, NMX Research and Solutions Inc., Canada
14:35-14:55 Title: Glucose Transporter (GLUTs) Inhibitors as Novel Anticancer Therapeutics

Dr. Xiaozhuo Chen, Associate Professor, Ohio University, USA

14:55-16:15

Title: NSP4: The Fourth Player at the Neutrophils Serine Proteases Table

Dr. Marcin Sienczyk, Assistant Professor, Wroclaw University of Science and Technology, Poland 

15:15-15:30 Coffee Break
15:30-15:50 Title: Discovery of Endonuclease Inhibitors - A New Class of Drugs to Combat Tissue Injury
Dr. Alexei G. Basnakian, Professor, University of Arkansas for Medical Sciences, USA
15:50-16:10

 

Title: Discovery of Novel Competitive GSK3 Beta Inhibitors for the Treatment of Mood Disorders
Dr. Angelo Reggiani, PI/Director, Department of Drug Discovery and Development, Italian Institute of Technology (IIT), Italy


16:10-16:30 Title: Scaffold Synthesis of Fluorescence Alkaloid Ageladine A, an Anticancer MMP-2 Inhibitor
Dr. Tomoko Mineno, Professor, Takasaki University of Health and Welfare, Japan
16:30-16:50 Title: Synthesis, Biological Evaluation and Molecular Modeling Study of Substituted Benzyl Benzamides as CETP Inhibitors
Dr. Reema Abu Khalaf, Associate Professor, Al-Zaytoonah University of Jordan, Jordan
16:50-17:10

 

Title: MERTK Promotes Wild-type EGFR NSCLCs Resistant to Irreversible EGFR TKIs

Dr. Dan Yan, Instructor, Emory University, USA
17:30-20:30 Welcome Banquet & Art Performance

© 2003-2018 All rights reserved by BITeomics Inc.
Contact Us: Tel: 0086-411-84799609, Fax: 0086-411-84796897